SCHEMBL7338142

SCHEMBL7338142

c1ccc(CN2CCN=C2CN(Cc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48
CYP2D6 P10635 3/20 0.48
TSHR P16473 3/20 0.48
CYP1A2 P05177 2/20 0.48
LMNA P02545 2/20 0.48
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
PDE6A P16499 1/20 0.48
ADRA2C P18825 1/20 0.48
MC4R P32245 1/20 0.48
ADRA1A P35348 1/20 0.48
HRH1 P35367 1/20 0.48
OPRM1 P35372 1/20 0.48
DRD3 P35462 1/20 0.48
MC3R P41968 1/20 0.48
SLC6A3 Q01959 1/20 0.48
KMT2A Q03164 1/20 0.48
PDE4D Q08499 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344251 0.91 HTR1D (0.44) HTR1DHTR1BCYP2D6TSHRCYP1A2
SCHEMBL7346849 0.87 NR1H2 (0.47) HTR1DHTR1BCYP2D6TSHRCYP1A2
SCHEMBL7337729 0.87 TSHR (0.50) HTR1DHTR1BCYP2D6TSHRCYP1A2
SCHEMBL7339207 0.85 CYP2D6 (0.49) HTR1DHTR1BCYP2D6TSHRCYP1A2
SCHEMBL7338899 0.83 TSHR (0.44) HTR1DHTR1BCYP2D6TSHRCYP1A2
SCHEMBL7345751 0.83 CYP2D6 (0.47) HTR1DHTR1BCYP2D6TSHRCYP1A2
SCHEMBL7344285 0.82 CYP2D6 (0.47) CYP2D6TSHRCYP1A2LMNAHTR1A
SCHEMBL7339633 0.81 CYP1A2 (0.46) CYP2D6TSHRCYP1A2LMNAHTR1A
SCHEMBL7337002 0.80 CYP1A2 (0.45) CYP2D6TSHRCYP1A2LMNAHTR1A
SCHEMBL7344115 0.80 CYP1A2 (0.45) CYP2D6TSHRCYP1A2LMNAHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0598962-B1 Imidazole derivatives as calcium channel blockers NEUROSEARCH AS (DK) 1999-02-17 EP claimed
EP-0598962-A1 Imidazole derivatives as calcium channel blockers NEUROSEARCH A/S (DK) 1994-06-01 EP claimed
US-5296493-A Analgesics or antiischemics NEUROSEARCH A/S (DK) 1994-03-22 US claimed
EP-0598962-B1 Imidazole derivatives as calcium channel blockers NEUROSEARCH AS (DK) 1999-02-17 EP disclosed
EP-0598962-A1 Imidazole derivatives as calcium channel blockers NEUROSEARCH A/S (DK) 1994-06-01 EP disclosed
US-5296493-A Analgesics or antiischemics NEUROSEARCH A/S (DK) 1994-03-22 US disclosed