SCHEMBL7338573

SCHEMBL7338573

CCCC(=O)Oc1ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)OC)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.50
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
CTSS P25774 6/20 0.46
CTSK P43235 5/20 0.46
ACE P12821 1/20 0.46
PPARG P37231 2/20 0.45
PPARA Q07869 2/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
ABCB1 P08183 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
CACNA1B Q00975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1972111 0.86 KLK5 (0.54) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL5408855 0.84 PPARG (0.57) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL5408845 0.84 PPARG (0.57) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL4937975 0.84 ITGB3 (0.61) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL4937967 0.84 ITGB3 (0.61) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL16815979 0.84 ITGB3 (0.64) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL15593763 0.84 ITGB3 (0.64) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL2802881 0.84 KLK5 (0.52) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL2802882 0.84 KLK5 (0.52) KLK5ITGB3ITGA2BCTSSCTSK
SCHEMBL22604385 0.83 GAA (0.60) KLK5ITGB3ITGA2BCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767792-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
US-5977101-A Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity SMITHKLINE BEECHAM CORPORATION (US) 1999-11-02 US disclosed
EP-0767792-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-04-16 EP disclosed
WO-1996000730-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-01-11 WO disclosed