SCHEMBL7339679

SCHEMBL7339679

OC1CCC2(CC1)CCC(/C=N/Nc1ncc[nH]1)CC2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR2C P28335 1/20 0.36
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 1/20 0.32
ATP1A1 P05023 2/20 0.31
ATP1B1 P05026 2/20 0.31
ATP1A3 P13637 2/20 0.31
ATP1B2 P14415 2/20 0.31
ATP1A2 P50993 2/20 0.31
ATP1B3 P54709 2/20 0.31
FXYD2 P54710 2/20 0.31
ATP1A4 Q13733 2/20 0.31
FDPS P14324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339687 1.00 GAA (0.39) GAAMAPTL3MBTL1HTR1AHTR1D
SCHEMBL7338313 0.88 GAA (0.36) GAAMAPTL3MBTL1HTR1AHTR1D
SCHEMBL7338321 0.88 GAA (0.36) GAAMAPTL3MBTL1HTR1AHTR1D
SCHEMBL7339639 0.78 GAA (0.33) GAAMAPTL3MBTL1HTR1AHTR1D
SCHEMBL7341962 0.77 GAA (0.35) GAAMAPTL3MBTL1
SCHEMBL7340876 0.75 ATP1A1 (0.47) HTR1AATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL7340871 0.75 ATP1A1 (0.47) HTR1AATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL7345767 0.67 GAA (0.31) GAAMAPTL3MBTL1ALDH1A1
SCHEMBL7346834 0.64 ATP1A1 (0.40) GAAALDH1A1KMT2AATP1A1ATP1B1
SCHEMBL7346837 0.64 ATP1A1 (0.40) GAAALDH1A1KMT2AATP1A1ATP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0578080-B1 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same SIGMA TAU IND FARMACEUTI (IT) 1997-04-23 EP claimed
EP-0578080-A2 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1994-01-12 EP claimed
EP-0578080-B1 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same SIGMA TAU IND FARMACEUTI (IT) 1997-04-23 EP disclosed
US-5444082-A Treats hypertension and heart failure SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 1995-08-22 US disclosed
EP-0578080-A2 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1994-01-12 EP disclosed