SCHEMBL7340523

SCHEMBL7340523

CC[C@H](C)[C@H](NC(=O)N(C)Cc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)N(C)Cc1ccccn1)[C@@H](C)CC

nearest known ligand 0.85

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.85
REN P00797 9/20 0.47
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
CTSD P07339 7/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333171 1.00 CA2 (0.85) CA2RENCYP1A2CYP2D6MAPT
SCHEMBL7341313 1.00 CA2 (0.85) CA2RENCYP1A2CYP2D6MAPT
A-77003 SCHEMBL8749867 0.92 CA2 (1.00) CA2CYP1A2CYP2D6MAPTTSHR
A-77003 SCHEMBL7337518 0.92 CA2 (1.00) CA2CYP1A2CYP2D6MAPTTSHR
A-77003 SCHEMBL2770013 0.92 CA2 (1.00) CA2CYP1A2CYP2D6MAPTTSHR
A-76928 SCHEMBL6449595 0.92 CA2 (1.00) CA2CYP1A2CYP2D6MAPTTSHR
A-77003 SCHEMBL6448973 0.92 CA2 (1.00) CA2CYP1A2CYP2D6MAPTTSHR
SCHEMBL7278095 0.90 CA2 (0.96) CA2CYP1A2CYP2D6MAPTTSHR
SCHEMBL7305188 0.89 CA2 (0.87) CA2RENCYP2D6MAPTCYP3A4
SCHEMBL7341491 0.87 CA2 (0.89) CA2CYP1A2CYP2D6MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed