SCHEMBL7340722

SCHEMBL7340722

CC(C)[C@H](NC(=O)N(C)Cc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.83

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.83
KLK5 Q9Y337 1/20 0.49
REN P00797 3/20 0.48
BACE1 P56817 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
PSEN1 P49768 4/20 0.48
PSEN2 P49810 4/20 0.48
APH1B Q8WW43 4/20 0.48
NCSTN Q92542 4/20 0.48
APH1A Q96BI3 4/20 0.48
PSENEN Q9NZ42 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7331805 1.00 CA2 (0.83) CA2KLK5RENBACE1CYP1A2
SCHEMBL7332653 1.00 CA2 (0.83) CA2KLK5RENBACE1CYP1A2
A-77003 SCHEMBL2770013 0.91 CA2 (1.00) CA2BACE1CYP1A2CYP3A4CYP2D6
A-77003 SCHEMBL6448973 0.91 CA2 (1.00) CA2BACE1CYP1A2CYP3A4CYP2D6
A-76928 SCHEMBL6449595 0.91 CA2 (1.00) CA2BACE1CYP1A2CYP3A4CYP2D6
A-77003 SCHEMBL7337518 0.91 CA2 (1.00) CA2BACE1CYP1A2CYP3A4CYP2D6
A-77003 SCHEMBL8749867 0.91 CA2 (1.00) CA2BACE1CYP1A2CYP3A4CYP2D6
SCHEMBL7332468 0.90 CA2 (0.83) CA2KLK5BACE1CYP3A4CYP2D6
SCHEMBL7306151 0.90 CA2 (0.83) CA2BACE1CYP3A4CYP2D6CYP2C19
SCHEMBL7343854 0.89 CA2 (0.71) CA2RENCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed