SCHEMBL7343283

SCHEMBL7343283

CC(C[CH]C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)NCc1ccncc1)C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
CYP3A4 P08684 1/20 0.50
KLKB1 P03952 6/20 0.48
MMP9 P14780 2/20 0.47
MMP8 P22894 2/20 0.47
PPARG P37231 2/20 0.47
KLK1 P06870 1/20 0.46
CTSL P07711 1/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
MME P08473 1/20 0.44
ACE P12821 1/20 0.44
CPA1 P15085 1/20 0.44
ACE2 Q9BYF1 1/20 0.44
PSMB1 P20618 1/20 0.44
PSMB9 P28065 1/20 0.44
PSMB5 P28074 1/20 0.44
PSMB10 P40306 1/20 0.44
PSMB2 P49721 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337025 0.95 KLKB1 (0.52) KLKB1MMP9MMP8PPARGMME
SCHEMBL7339080 0.91 KLKB1 (0.58) KLKB1KLK1
SCHEMBL7346201 0.87 PPARG (0.48) KLKB1MMP9MMP8PPARGKLK1
SCHEMBL7343062 0.87 KLKB1 (0.47) KLKB1MMP9MMP8PPARGKLK1
SCHEMBL7341933 0.86 PPARG (0.50) CYP3A4MMP9MMP8PPARGCTSS
SCHEMBL7345736 0.86 REN (0.51) KLKB1MMP9MMP8PPARGCTSL
SCHEMBL7348629 0.86 PPARG (0.47) ALDH1A1KLKB1MMP9MMP8PPARG
SCHEMBL7344073 0.85 PPARG (0.62) MMP9MMP8PPARGMMEACE
SCHEMBL7340612 0.85 PPARG (0.47) KLKB1MMP9MMP8PPARGCTSL
SCHEMBL7341957 0.84 PLG (0.50) MMP9MMP8PPARGMMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed