SCHEMBL7344442

SCHEMBL7344442

CC(C)[C@H](NC(=O)C=Cc1ccncc1)C(=O)N[C@@H](Cc1ccccc1)C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)C=Cc1ccncc1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.52
BACE1 P56817 12/20 0.50
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPT P10636 1/20 0.45
CTSD P07339 1/20 0.45
NOS2 P35228 3/20 0.43
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344438 1.00 CA2 (0.52) CA2BACE1ALDH1A1CYP1A2CYP3A4
SCHEMBL7311439 0.89 NAMPT (0.50) CA2BACE1ALDH1A1CYP1A2CYP3A4
SCHEMBL7311433 0.89 NAMPT (0.50) CA2BACE1ALDH1A1CYP1A2CYP3A4
SCHEMBL7307928 0.87 CA2 (0.52) CA2BACE1ALDH1A1CYP1A2CYP3A4
SCHEMBL7333725 0.87 CA2 (0.52) CA2BACE1ALDH1A1CYP1A2CYP3A4
SCHEMBL7342544 0.85 CA2 (0.59) CA2BACE1CYP1A2MAPTCTSD
SCHEMBL7342550 0.85 CA2 (0.59) CA2BACE1CYP1A2MAPTCTSD
SCHEMBL6452553 0.83 CA2 (0.62) CA2BACE1CYP1A2MAPTCTSD
SCHEMBL7277346 0.81 CA2 (0.56) CA2BACE1MAPK1CTSD
SCHEMBL7307580 0.80 CA2 (0.53) CA2BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed