SCHEMBL7346302

SCHEMBL7346302

COc1c(N)c2ccccc2oc1=O

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 8/20 0.62
KDM4E B2RXH2 6/20 0.62
ALDH1A1 P00352 3/20 0.62
CA12 O43570 1/20 0.56
CA9 Q16790 1/20 0.56
MAPT P10636 3/20 0.55
MGAM O43451 3/20 0.52
SI P14410 3/20 0.52
MGAM2 Q2M2H8 3/20 0.52
LMNA P02545 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.51
POLB P06746 2/20 0.51
CYP2C9 P11712 2/20 0.50
HSD17B10 Q99714 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14638270 0.86 GAA (0.62) GAAKDM4EALDH1A1CA12CA9
SCHEMBL29854772 0.84 CA12 (0.66) GAAKDM4EALDH1A1CA12CA9
SCHEMBL831768 0.84 CA12 (0.66) GAAKDM4EALDH1A1CA12CA9
SCHEMBL2266790 0.81 CA12 (0.58) KDM4EALDH1A1CA12CA9MAPT
SCHEMBL9528397 0.79 KDM4E (0.62) KDM4EALDH1A1CA12CA9MAPT
SCHEMBL15842594 0.79 CYP2C9 (0.57) GAAKDM4EALDH1A1CA12CA9
SCHEMBL1230426 0.77 GAA (1.00) GAAKDM4EALDH1A1MAPTMGAM
SCHEMBL94134 0.77 GAA (0.69) GAAKDM4EALDH1A1MAPTMGAM
SCHEMBL17760847 0.76 CA12 (0.60) GAAKDM4EALDH1A1CA12CA9
SCHEMBL22193185 0.76 POLB (0.62) GAAKDM4EALDH1A1MAPTMGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542708-B1 Substituted beta-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2001-05-30 EP disclosed
US-5973003-A TREATMENT OF THROMBOSIS, STROKE, MYOCARDIAL INFARCTION, INFLAMMATION AND ARTERIOSCLEROSIS G. D. SEARLE & CO. (US) 1999-10-26 US disclosed
US-5703125-A MELT BLEND OF SOAP, SURFACTANT AND SOLVENT G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
EP-0614360-B1 SUBSTITUTED BETA-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1997-03-19 EP disclosed
EP-0614360-A1 SUBSTITUTED -g(b)-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS. SEARLE & CO (US) 1994-09-14 EP disclosed
US-5344957-A Amidinoiphenyl-substituted G.D. SEARLE & CO. (US) 1994-09-06 US disclosed
EP-0542708-A1 Substituted B-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-05-19 EP disclosed
WO-1993007867-A1 SUBSTITUTED β-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-04-29 WO disclosed