SCHEMBL7346337

SCHEMBL7346337

CCC(CC)(C(=O)O)C(CCC(=O)O)NC(=O)CCC(=O)Nc1ccc(C=NN)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
ITGB3 P05106 6/20 0.38
ITGA2B P08514 6/20 0.38
CYP1A1 P04798 1/20 0.37
KMT2A Q03164 3/20 0.36
POLB P06746 2/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353903 0.94 CA12 (0.37) CA12CA1CA2CA4CA9
SCHEMBL7346305 0.81 ITGB3 (0.59) ITGB3ITGA2B
SCHEMBL7346087 0.81 ITGB3 (0.53) CA12CA1CA2CA4CA9
SCHEMBL7423763 0.80 ITGB3 (0.44) CA12CA1CA2CA4CA9
SCHEMBL6980785 0.78 CA12 (0.59) CA12CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL6983894 0.77 CA12 (0.57) CA12CA1CA2CA4CA9
SCHEMBL7348197 0.76 ITGB3 (0.63) CA12CA1CA2CA4CA9
SCHEMBL7353870 0.76 ITGB3 (0.57) ITGB3ITGA2B
SCHEMBL7345488 0.76 ITGB3 (0.54) CA12CA1CA2CA4CA9
SCHEMBL7346326 0.75 ITGB3 (0.39) CA12CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542708-B1 Substituted beta-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2001-05-30 EP disclosed
US-5973003-A TREATMENT OF THROMBOSIS, STROKE, MYOCARDIAL INFARCTION, INFLAMMATION AND ARTERIOSCLEROSIS G. D. SEARLE & CO. (US) 1999-10-26 US disclosed
EP-0614360-B1 SUBSTITUTED BETA-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1997-03-19 EP disclosed
US-5344957-A Amidinoiphenyl-substituted G.D. SEARLE & CO. (US) 1994-09-06 US disclosed
US-5239113-A Anticoagulants MONSANTO COMPANY (US) 1993-08-24 US disclosed
EP-0542708-A1 Substituted B-amino acid derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-05-19 EP disclosed
WO-1993007867-A1 SUBSTITUTED β-AMINO ACID DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-04-29 WO disclosed