SCHEMBL7347239

SCHEMBL7347239

COc1ccc2sc(-c3ccc(O)cc3)cc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.58
HDAC6 Q9UBN7 1/20 0.58
ESR2 Q92731 4/20 0.54
ESR1 P03372 3/20 0.54
BACE1 P56817 1/20 0.53
CLK1 P49759 2/20 0.47
DYRK1A Q13627 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
SULT1A1 P50225 1/20 0.47
CA2 P00918 1/20 0.47
ABL1 P00519 2/20 0.46
ABCB1 P08183 2/20 0.46
BCR P11274 2/20 0.46
HSP90AA1 P07900 1/20 0.45
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171301 0.88 ESR2 (0.68) APPHDAC6ESR2ESR1SULT1A1
SCHEMBL9151832 0.84 BACE1 (0.56) HDAC6ESR2ESR1BACE1CLK1
SCHEMBL23815138 0.81 ESR1 (0.72) APPESR2ESR1CLK1DYRK1A
SCHEMBL498648 0.81 ESR2 (0.73) APPHDAC6ESR2ESR1SULT1A1
SCHEMBL21014552 0.79 HDAC6 (0.49) APPHDAC6BACE1CLK1DYRK1A
SCHEMBL1179171 0.77 HDAC6 (0.60) HDAC6CLK1DYRK1ADYRK1BNPC1
SCHEMBL1665299 0.77 NPC1 (0.56) APPHDAC6ESR2ESR1CA2
SCHEMBL31310542 0.77 NPC1 (0.56) APPHDAC6ESR2ESR1CA2
SCHEMBL7349045 0.76 FFAR4 (0.58) HDAC6CLK1DYRK1ADYRK1BALDH1A1
SCHEMBL6173418 0.76 RAB9A (0.68) APPHDAC6CA2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993300-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2002-07-31 EP disclosed
US-6284756-B1 ANTICOAGULANT ELI LILLY AND COMPANY 2001-09-04 US disclosed
EP-0993300-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-04-19 EP disclosed
WO-1998048798-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed