SCHEMBL7347756

SCHEMBL7347756

Cc1c(-c2ccc(O[Si](C(C)C)(C(C)C)C(C)C)cc2)sc2cc(OC(C)C)cc(Nc3ccc(OCCN4CCCC4)cc3)c12

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.40
ESR2 Q92731 11/20 0.40
ITGA4 P13612 1/20 0.39
SRC P12931 2/20 0.39
ENPP3 O14638 1/20 0.39
ENPP1 P22413 1/20 0.38
FLT3 P36888 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346989 0.94 ESR1 (0.44) ESR1ESR2ITGA4ENPP3
SCHEMBL7352553 0.90 ESR1 (0.49) ESR1ESR2
SCHEMBL7352615 0.87 ITGA4 (0.45) ESR1ESR2ITGA4SRCFLT3
SCHEMBL7438752 0.84 ESR1 (0.49) ESR1ESR2ENPP3ENPP1
SCHEMBL7349173 0.81 ESR1 (0.55) ESR1ESR2
SCHEMBL7347006 0.78 ITGA4 (0.53) ESR1ESR2ITGA4SRC
SCHEMBL7348137 0.76 ESR1 (0.55) ESR1ESR2ENPP3
SCHEMBL7347763 0.75 ESR1 (0.49) ESR1ESR2ENPP3ENPP1
SCHEMBL7350932 0.73 ESR1 (0.62) ESR1ESR2
SCHEMBL7772332 0.70 ESR1 (0.74) ESR1ESR2ENPP3ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997460-B1 Benzothiophene compounds as antithrombotic agents and intermediates LILLY CO ELI (US) 2002-12-11 EP disclosed
US-6133262-A 3-AMINOBENZO(B)THIOPHENE DERIVATIVES ELI LILLY AND COMPANY (US) 2000-10-17 US disclosed
EP-0997460-A1 Benzothiophene compounds as antithrombotic agents and intermediates ELI LILLY AND COMPANY (US) 2000-05-03 EP disclosed