SCHEMBL7348263

SCHEMBL7348263

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2C(=O)c3ccccc3C2=O)C1c1ccccc1Cl

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.66
KDM4E B2RXH2 4/20 0.57
CYP2C9 P11712 3/20 0.57
TBXA2R P21731 3/20 0.57
ADRA1A P35348 3/20 0.57
SLC6A3 Q01959 3/20 0.57
ABCB11 O95342 3/20 0.57
CYP3A4 P08684 3/20 0.57
GAA P10253 3/20 0.57
ALDH1A1 P00352 3/20 0.57
MEN1 O00255 2/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2C19 P33261 2/20 0.57
KMT2A Q03164 2/20 0.57
HIF1A Q16665 2/20 0.57
ABCB1 P08183 2/20 0.57
ADORA3 P0DMS8 2/20 0.57
ADRB3 P13945 2/20 0.57
OPRK1 P41145 2/20 0.57
SCN5A Q14524 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9673018 0.93 CYP2C9 (0.68) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL7342557 0.88 HSD17B10 (0.66) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL7344861 0.88 HSD17B10 (0.66) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL5474815 0.87 ABCB11 (0.67) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL4986252 0.86 TBXA2R (0.75) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL3185862 0.86 TBXA2R (0.75) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL31473037 0.86 TBXA2R (0.75) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL9673483 0.86 HSD17B10 (0.63) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL7350118 0.86 HSD17B10 (0.61) HSD17B10KDM4ECYP2C9TBXA2RADRA1A
SCHEMBL7347116 0.86 HSD17B10 (0.56) HSD17B10CYP2C9ADRA1ASLC6A3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed