SCHEMBL7348386

SCHEMBL7348386

N=C(N)Nc1cccc(C(=O)NCC(=O)Nc2cccc3ccc(CCC(=O)O)cc23)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.48
ITGA2B P08514 2/20 0.48
TAOK1 Q7L7X3 1/20 0.45
ITGB1 P05556 3/20 0.45
ITGAV P06756 3/20 0.45
MDM4 O15151 2/20 0.45
ITGA5 P08648 2/20 0.45
MDM2 Q00987 2/20 0.45
TRPV1 Q8NER1 4/20 0.43
RXFP1 Q9HBX9 1/20 0.42
SIRT1 Q96EB6 1/20 0.41
ITGB5 P18084 1/20 0.41
PPARG P37231 1/20 0.41
NR1H4 Q96RI1 2/20 0.40
PPARD Q03181 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
F2 P00734 2/20 0.40
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348423 0.88 ITGB3 (0.45) ITGB3ITGA2BTAOK1ITGB1ITGAV
SCHEMBL7346500 0.86 ITGB3 (0.60) ITGB3ITGA2BITGB1ITGAVRXFP1
SCHEMBL6778210 0.85 ITGB3 (0.45) ITGB3ITGA2BTAOK1ITGB1ITGAV
SCHEMBL7337027 0.83 RXFP1 (0.43) ITGB3ITGA2BITGB1ITGAVMDM4
SCHEMBL7348081 0.82 ITGB3 (0.43) ITGB3ITGA2BITGB1ITGAVMDM4
SCHEMBL7348024 0.81 ITGB3 (0.42) ITGB3ITGA2BITGB1ITGAVMDM4
SCHEMBL7340337 0.80 ITGB3 (0.41) ITGB3ITGA2BITGB1ITGAVMDM4
SCHEMBL6777380 0.79 SMN1; SMN2 (0.44) ITGB3ITGA2BITGB1ITGAVMDM4
SCHEMBL7340290 0.79 ITGB3 (0.42) ITGB3ITGA2BITGB1ITGAVMDM4
SCHEMBL7339868 0.79 RXFP1 (0.45) ITGB3TAOK1ITGB1ITGAVMDM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed