SCHEMBL7348998

SCHEMBL7348998

CCCCN1CCC(CCC(=O)c2cc(Cl)c(N)cc2OCc2cc(OC)cc(OC)c2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 9/20 0.77
ACHE P22303 6/20 0.77
MEN1 O00255 2/20 0.77
ALDH1A1 P00352 2/20 0.77
CYP2D6 P10635 2/20 0.77
KMT2A Q03164 2/20 0.77
CYP2C9 P11712 1/20 0.77
TSHR P16473 1/20 0.77
TP53 P04637 1/20 0.76
CYP3A4 P08684 1/20 0.76
CYP2C19 P33261 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7358076 0.99 HTR4 (0.76) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL7359859 0.97 HTR4 (0.77) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL7358480 0.97 HTR4 (0.75) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL7355077 0.93 MEN1 (0.70) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL7356578 0.90 MEN1 (0.76) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL7355573 0.89 MEN1 (0.69) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL549019 0.88 HTR4 (1.00) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL29604454 0.88 HTR4 (1.00) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL19961562 0.87 MEN1 (0.79) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL16058183 0.87 HTR4 (0.84) HTR4ACHEMEN1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-B1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX INC (US) 1998-09-23 EP disclosed
US-5763458-A NERVOUS SYSTEM DISORDERS, ANXIETY, ANTIDEPRESSANTS AND COGNITION ACTIVATORS SYNTEX (U.S.A.) INC. (US) 1998-06-09 US disclosed
WO-1994027965-A1 NOVEL 1-PHENYLALKANONE 5-HT4 RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1994-12-08 WO disclosed