SCHEMBL7349233

SCHEMBL7349233

N#Cc1cccc([C@@H]2CCCN(CCc3ccccc3)C2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 12/20 1.00
DRD2 P14416 12/20 1.00
CYP2D6 P10635 1/20 0.72
TSHR P16473 1/20 0.72
NFKB1 P19838 1/20 0.72
CASP1 P29466 1/20 0.72
NPSR1 Q6W5P4 1/20 0.71
DRD1 P21728 2/20 0.58
DRD4 P21917 2/20 0.58
DRD5 P21918 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7383021 0.93 DRD3 (1.00) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL7355118 0.84 DRD3 (1.00) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL7346180 0.84 DRD3 (1.00) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL872942 0.84 DRD3 (1.00) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL7351587 0.82 DRD3 (0.86) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL7380006 0.81 DRD3 (0.70) DRD3DRD2NFKB1DRD1DRD4
SCHEMBL10657469 0.81 DRD3 (0.70) DRD3DRD2NFKB1DRD1DRD4
SCHEMBL7349038 0.81 DRD3 (1.00) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL8844122 0.80 DRD2 (0.67) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL7351584 0.79 DRD2 (1.00) DRD3DRD2CYP2D6TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5594024-A ANTIDEPRESSANTS; TREATMENT OF NARCOLEPSY, SCHIZOPHRENIA, DRUG ABUSE THE UPJOHN COMPANY (US) 1997-01-14 US disclosed
US-5462947-A Nervous system disorders THE UPJOHN COMPANY (US) 1995-10-31 US disclosed
EP-0641320-A1 NEW CENTRALLY ACTING SUBSTITUTED PHENYLAZACYCLOALKANES PHARMACIA & UPJOHN COMPANY (US) 1995-03-08 EP disclosed
WO-1992018475-A2 SUBSTITUTED PHENYLAZACYCLOALKANES AS CNS AGENTS THE UPJOHN COMPANY (US) 1992-10-29 WO disclosed