SCHEMBL7349592

SCHEMBL7349592

CC([O])Sc1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
DDAH1 O94760 1/20 0.46
NOS1 P29475 1/20 0.46
LMNA P02545 4/20 0.41
POLB P06746 2/20 0.38
TSHR P16473 2/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
PTGS2 P35354 1/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
MAPT P10636 1/20 0.33
CHRM5 P08912 1/20 0.32
CHKA P35790 1/20 0.32
HPGD P15428 2/20 0.32
GAA P10253 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6095853 0.80 MEN1 (0.50) MEN1KMT2ADDAH1NOS1LMNA
Hydrochloric Acid SCHEMBL6097232 0.78 MEN1 (0.48) MEN1KMT2ADDAH1NOS1LMNA
SCHEMBL7349599 0.76 MEN1 (0.46) MEN1KMT2ADDAH1NOS1LMNA
SCHEMBL10402880 0.76 MEN1 (0.41) MEN1KMT2ADDAH1NOS1LMNA
SCHEMBL10402878 0.76 MEN1 (0.41) MEN1KMT2ADDAH1NOS1LMNA
SCHEMBL95521 0.75 LMNA (0.42) LMNAPOLBALDH1A1SMN1; SMN2MAOA
SCHEMBL5983975 0.73 HPGD (0.46) MEN1KMT2ALMNAPOLBALDH1A1
SCHEMBL7242681 0.73 MEN1 (0.42) MEN1KMT2ADDAH1NOS1LMNA
SCHEMBL7288566 0.71 HCAR2 (0.31)
SCHEMBL7123357 0.71 HSD17B10 (0.52) LMNATSHRALDH1A1SMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed