SCHEMBL7349743

SCHEMBL7349743

Cc1cc(C(=O)CCC(=O)O)c2c(c1)N(C)C(=O)CO2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
HTT P42858 2/20 0.41
TSHR P16473 1/20 0.41
HTR2A P28223 1/20 0.39
SLC6A4 P31645 1/20 0.39
HRH1 P35367 1/20 0.39
HTR3A P46098 1/20 0.39
PDE4D Q08499 1/20 0.39
KCNH2 Q12809 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP1A2 P05177 1/20 0.39
KMO O15229 1/20 0.37
POLB P06746 3/20 0.36
PLK1 P53350 1/20 0.34
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341338 0.87 PDE3B (0.42) PDE3BPDE3AKMT2AMEN1HTT
SCHEMBL7287945 0.84 PDE3B (0.49) PDE3BPDE3AHTTTSHRHTR2A
Hydrochloric Acid SCHEMBL7291531 0.83 PDE3B (0.48) PDE3BPDE3AHTTTSHRHTR2A
SCHEMBL7291509 0.80 PDE3B (0.48) PDE3BPDE3AKMT2AMEN1HTT
SCHEMBL22919064 0.80 PDE3B (0.48) PDE3BPDE3AHTTTSHRHTR2A
SCHEMBL10267004 0.74 PDE3B (0.52) PDE3BPDE3AKMT2AMEN1HTT
SCHEMBL7350571 0.73 PDE3B (0.45) PDE3BPDE3AKMT2AMEN1HTT
SCHEMBL10642537 0.72 PDE3B (0.42) PDE3BPDE3AHTTTSHRHTR2A
SCHEMBL7341783 0.72 PDE3B (0.40) PDE3BPDE3AHTTTSHRHTR2A
SCHEMBL4968297 0.72 KMO (0.52) KMT2AMEN1HTTTSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081242-A Cardiotonic and bronchodilator agents; phosphodiesterase inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1992-01-14 US disclosed
US-4766118-A CARDIOTONIC AGENTS, PHOSPHODIESTERASE INHIBITORS ORTHO PHARMACEUTICAL CORPORATION (US) 1988-08-23 US disclosed
EP-0272914-A2 6-Benzoxazinyl- and 6-benzothiazinyl-2,3,4,5-tetrahydropyridazin-3-ones ORTHO PHARMACEUTICAL CORPORATION (US) 1988-06-29 EP disclosed
US-4721784-A MUSCLE RELAXANTS, BRONCHODILATOR AGENTS, CARDIOTONIC AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1988-01-26 US disclosed