SCHEMBL7350997

SCHEMBL7350997

COc1ccc(OC)c(C2=CCOC2=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
KDM4E B2RXH2 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 3/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
ALOX12 P18054 1/20 0.43
RAB9A P51151 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP19A1 P11511 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30527909 0.81 L3MBTL1 (0.51) KDM4ETSHRALDH1A1MAPTHPGD
SCHEMBL2167797 0.76 BACE1 (0.52) KDM4EALDH1A1MAPTTDP1CYP19A1
SCHEMBL7351176 0.75 CYP19A1 (0.55) KDM4ESMN1; SMN2TSHRHTTALDH1A1
SCHEMBL9850097 0.75 NCOA1 (0.48) HDAC4HDAC8KDM4ESMN1; SMN2ALDH1A1
SCHEMBL196223 0.72 CA12 (0.68) HDAC4HDAC2HDAC8KDM4ESMN1; SMN2
SCHEMBL7349003 0.70 CYP19A1 (0.48) KDM4EALDH1A1MAPTHPGDCYP19A1
SCHEMBL10841088 0.70 HDAC4 (0.54) HDAC4HDAC2HDAC8KDM4ESMN1; SMN2
SCHEMBL16812904 0.68 HDAC4 (0.74) HDAC4HDAC2HDAC8KDM4ESMN1; SMN2
SCHEMBL5197914 0.68 CA12 (0.56) HDAC4HDAC2HDAC8KDM4ESMN1; SMN2
SCHEMBL16109474 0.68 HDAC4 (0.65) HDAC4HDAC2HDAC8KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027077-A1 2,1,3-BENZOTHIA(OXA)DIAZOLE DERIVATIVES AND THEIR USE AS ENDOTHELIN-RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-06-25 WO disclosed