SCHEMBL7351018

SCHEMBL7351018

O=c1oc2ccccc2c(O)c1C(CCc1ccccc1)Cc1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 5/20 0.61
CYP2C9 P11712 6/20 0.56
TOP1 P11387 1/20 0.55
VKORC1 Q9BQB6 3/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
ALB P02768 1/20 0.53
PCSK7 Q16549 1/20 0.53
HSD17B10 Q99714 1/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358731 0.90 NQO1 (0.65) NQO1CYP2C9TOP1VKORC1KDM4E
SCHEMBL7356247 0.88 NQO1 (0.76) NQO1CYP2C9VKORC1KDM4EALDH1A1
SCHEMBL7354054 0.88 NQO1 (0.67) NQO1CYP2C9VKORC1KDM4EALDH1A1
SCHEMBL7352699 0.85 CYP2C9 (0.69) NQO1CYP2C9TOP1VKORC1KDM4E
SCHEMBL7354556 0.85 CYP2C9 (0.69) NQO1CYP2C9TOP1VKORC1KDM4E
SCHEMBL4294895 0.84 NQO1 (0.65) NQO1CYP2C9VKORC1KDM4EALDH1A1
SCHEMBL7356446 0.82 CYP2C9 (0.72) NQO1CYP2C9TOP1VKORC1KDM4E
SCHEMBL9210173 0.82 NQO1 (0.61) NQO1CYP2C9VKORC1ALDH1A1PCSK7
SCHEMBL14033878 0.82 VKORC1 (0.71) NQO1CYP2C9VKORC1KDM4EALDH1A1
SCHEMBL7358027 0.81 NQO1 (0.64) NQO1CYP2C9VKORC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682663-B1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS UPJOHN CO (US) 2001-04-18 EP claimed
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US claimed
EP-0682663-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-22 EP claimed
WO-1994018188-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL[B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS THE UPJOHN COMPANY (US) 1994-08-18 WO claimed
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
EP-0682663-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-22 EP disclosed
WO-1994018188-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL[B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS THE UPJOHN COMPANY (US) 1994-08-18 WO disclosed