SCHEMBL7355223

SCHEMBL7355223

CC1CC(=O)c2c(OCc3ccccc3)ccc(-c3ccccn3)c2C1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 8/20 0.61
GABRB3 P28472 8/20 0.61
GABRA5 P31644 8/20 0.61
GABRA1 P14867 7/20 0.61
GABRA3 P34903 7/20 0.61
GABRA2 P47869 7/20 0.61
MAOA P21397 2/20 0.39
GRM5 P41594 1/20 0.38
FBP1 P09467 1/20 0.38
MAOB P27338 1/20 0.37
BRD4 O60885 3/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
ABCG2 Q9UNQ0 2/20 0.36
CREBBP Q92793 1/20 0.36
CSNK2A2 P19784 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356851 0.80 GABRG2 (0.78) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7360811 0.79 GABRG2 (0.71) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7353297 0.76 GABRG2 (1.00) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7356856 0.76 GABRG2 (1.00) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7358466 0.76 GABRG2 (0.77) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7358004 0.74 GABRG2 (0.64) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7357419 0.73 GABRG2 (0.67) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7351990 0.73 GABRG2 (0.78) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7349798 0.73 GABRG2 (0.78) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7355669 0.72 GABRG2 (0.77) GABRG2GABRB3GABRA5GABRA1GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156761-A Substituted tetralone derivatives for enhancing cognition MERCK SHARPE & DOHME LIMITED (GB) 2000-12-05 US disclosed