SCHEMBL7355405

SCHEMBL7355405

COc1ccc(C(F)(F)F)cc1NC(=O)C(O)[C@H](N)CC1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 15/20 0.53
METAP1 P53582 6/20 0.48
CTSD P07339 2/20 0.46
KCNT1 Q5JUK3 1/20 0.44
KCNT2 Q6UVM3 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7356397 0.99 METAP2 (0.52) METAP2METAP1CTSDKCNT1KCNT2
SCHEMBL7359948 0.91 METAP2 (0.54) METAP2METAP1LMNA
Hydrochloric Acid SCHEMBL7355342 0.90 METAP2 (0.53) METAP2METAP1LMNA
SCHEMBL7362128 0.86 METAP2 (0.56) METAP2METAP1
SCHEMBL7360124 0.86 METAP2 (0.57) METAP2METAP1
Hydrochloric Acid SCHEMBL7353700 0.85 METAP2 (0.55) METAP2METAP1
Hydrochloric Acid SCHEMBL7352300 0.85 METAP2 (0.56) METAP2METAP1
SCHEMBL7355934 0.85 KMT2A (0.58) METAP2METAP1TDP1LMNA
Hydrochloric Acid SCHEMBL7352804 0.84 KMT2A (0.57) METAP2METAP1LMNA
SCHEMBL7360902 0.83 METAP2 (0.59) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed