SCHEMBL7356331

SCHEMBL7356331

COC(=O)[C@@H](N)Cc1ccc(NC(=O)c2cccnc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.64
SMN1; SMN2 Q16637 4/20 0.64
NPC1 O15118 3/20 0.64
TP53 P04637 2/20 0.57
ALDH1A1 P00352 3/20 0.56
NPSR1 Q6W5P4 2/20 0.56
MAPT P10636 3/20 0.55
GFER P55789 1/20 0.55
ROCK2 O75116 1/20 0.54
ROCK1 Q13464 1/20 0.54
GAA P10253 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
KMT2A Q03164 3/20 0.53
CYP3A4 P08684 1/20 0.53
LMNA P02545 1/20 0.52
HIF1A Q16665 1/20 0.52
MEN1 O00255 2/20 0.52
TSHR P16473 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27573780 0.99 RAB9A (0.62) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
Hydrochloric Acid SCHEMBL7356325 0.99 RAB9A (0.62) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
SCHEMBL5607137 0.87 RAB9A (0.64) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
SCHEMBL5607141 0.87 RAB9A (0.64) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
SCHEMBL27505713 0.85 GAA (0.56) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
SCHEMBL5164978 0.85 GAA (0.56) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
Hydrochloric Acid SCHEMBL7350429 0.84 GAA (0.55) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
Hydrochloric Acid SCHEMBL27553335 0.84 GAA (0.55) RAB9ASMN1; SMN2NPC1TP53ALDH1A1
Hydrochloric Acid SCHEMBL7358984 0.84 NPC1 (0.54) RAB9ASMN1; SMN2NPC1ALDH1A1MAPT
SCHEMBL22982998 0.80 RAB9A (0.73) RAB9ASMN1; SMN2NPC1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140792-A1 3,4-DIAMINO-3-CYCLOBUTENE-1,2-DIONE DERIVATIVES WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-10 EP disclosed
US-6166050-A 3,4-diamino-3-cyclobutene-1,2-dione derivatives which inhibit leukocyte adhesion mediated by VLA-4 AMERICAN HOME PRODUCTS CORPORATION (US) 2000-12-26 US disclosed
WO-2000035855-A1 3,4-DIAMINO-3-CYCLOBUTENE-1,2-DIONE DERIVATIVES WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-22 WO disclosed