SCHEMBL7357932

SCHEMBL7357932

O=c1oc2c(c(O)c1Cc1ccccc1)CCCC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 12/20 0.64
KDM4E B2RXH2 3/20 0.47
MAPT P10636 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
VKORC1 Q9BQB6 4/20 0.47
GAA P10253 2/20 0.45
MAPK1 P28482 2/20 0.45
JAK2 O60674 1/20 0.45
POLB P06746 1/20 0.45
PKM P14618 1/20 0.45
MPI P34949 1/20 0.45
HTT P42858 1/20 0.45
BLM P54132 1/20 0.45
MCL1 Q07820 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SHBG P04278 1/20 0.43
GLA P06280 1/20 0.42
HSD17B3 P37058 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ERAP1 Q9NZ08 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354114 0.99 NQO1 (0.63) NQO1KDM4EMAPTRXFP1VKORC1
SCHEMBL7357697 0.99 NQO1 (0.63) NQO1KDM4EMAPTRXFP1VKORC1
SCHEMBL7356934 0.99 NQO1 (0.63) NQO1KDM4EMAPTRXFP1VKORC1
SCHEMBL7350101 0.99 NQO1 (0.63) NQO1KDM4EMAPTRXFP1VKORC1
SCHEMBL7357238 0.99 NQO1 (0.63) NQO1KDM4EMAPTRXFP1VKORC1
SCHEMBL11161693 0.97 NQO1 (0.61) NQO1KDM4EMAPTRXFP1VKORC1
SCHEMBL9212226 0.83 NQO1 (0.47) NQO1GAAPKMSMN1; SMN2MEN1
SCHEMBL9204534 0.82 NQO1 (0.45) NQO1KDM4EMAPTGAAMAPK1
SCHEMBL7379070 0.78 NQO1 (0.45) NQO1KDM4EMAPTVKORC1GAA
SCHEMBL7358110 0.77 NQO1 (0.44) NQO1KDM4EMAPTVKORC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0682663-B1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS UPJOHN CO (US) 2001-04-18 EP disclosed
US-6169181-B1 HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITORS PHARMACIA & UPJOHN COMPANY 2001-01-02 US disclosed
US-5852195-A Pyranone compounds useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1998-12-22 US disclosed
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed
EP-0682663-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-22 EP disclosed
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed
WO-1994018188-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL[B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS THE UPJOHN COMPANY (US) 1994-08-18 WO disclosed
US-4418142-A ALDEHYDE SCAVANGERS AGFA GEVAERT AKTIENGESELLSCHAFT (DE) 1983-11-29 US disclosed
EP-0049449-B1 PHOTOSENSITIVE PHOTOGRAPHIC RECORDING MATERIAL BASED ON SILVER HALIDE Agfa-Gevaert AG (DE) 1983-09-28 EP disclosed
EP-0049449-A1 Photosensitive photographic recording material based on silver halide Agfa-Gevaert AG (DE) 1982-04-14 EP disclosed