SCHEMBL7357953

SCHEMBL7357953

COc1ccc(CNc2ccccc2Cl)cc1OC1CCOC1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 12/20 0.50
PDE4A P27815 9/20 0.50
PDE4B Q07343 8/20 0.50
PDE4C Q08493 7/20 0.50
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
UTS2R Q9UKP6 1/20 0.44
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
JAK3 P52333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL69444 0.86 PDE4D (0.60) PDE4DPDE4APDE4BPDE4CKDM4E
SCHEMBL7793212 0.80 MAPT (0.68) PDE4DKDM4EALDH1A1LMNAMAPT
SCHEMBL7361002 0.78 PDE4D (0.62) PDE4DPDE4APDE4BPDE4C
SCHEMBL7357379 0.78 PDE4D (0.76) PDE4DPDE4APDE4BPDE4C
SCHEMBL7358488 0.78 KMT2A (0.56) PDE4DPDE4APDE4BPDE4CALDH1A1
SCHEMBL12013392 0.76 PDE4D (0.45) PDE4DPDE4APDE4BPDE4C
SCHEMBL7149759 0.73 PDE4D (0.54) PDE4DPDE4APDE4BPDE4C
SCHEMBL7353005 0.72 PDE4D (0.48) PDE4DPDE4APDE4BPDE4C
SCHEMBL7353099 0.72 PDE4D (0.60) PDE4DPDE4APDE4BPDE4C
SCHEMBL1157245 0.71 PDE4D (0.48) PDE4DPDE4APDE4BPDE4CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741707-B1 SUBSTITUTED AROMATIC COMPOUNDS AS c.AMP PHOSPHODIESTERASE- AND TNF-INHIBITORS RHONE POULENC RORER LTD (GB) 1998-04-01 EP claimed
EP-0741707-A1 SUBSTITUTED AROMATIC COMPOUNDS AS c.AMP PHOSPHODIESTERASE- AND TNF-INHIBITORS RHONE-POULENC RORER LIMITED (GB) 1996-11-13 EP claimed
WO-1995020578-A1 SUBSTITUTED AROMATIC COMPOUNDS AS c.AMP PHOSPHODIESTERASE- AND TNF-INHIBITORS RHONE-POULENC RORER LIMITED (GB) 1995-08-03 WO claimed
EP-0741707-B1 SUBSTITUTED AROMATIC COMPOUNDS AS c.AMP PHOSPHODIESTERASE- AND TNF-INHIBITORS RHONE POULENC RORER LTD (GB) 1998-04-01 EP disclosed
EP-0741707-A1 SUBSTITUTED AROMATIC COMPOUNDS AS c.AMP PHOSPHODIESTERASE- AND TNF-INHIBITORS RHONE-POULENC RORER LIMITED (GB) 1996-11-13 EP disclosed
WO-1995020578-A1 SUBSTITUTED AROMATIC COMPOUNDS AS c.AMP PHOSPHODIESTERASE- AND TNF-INHIBITORS RHONE-POULENC RORER LIMITED (GB) 1995-08-03 WO disclosed