SCHEMBL7357997

SCHEMBL7357997

Cc1cccc(C#N)c1CN

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.54
LOXL2 Q9Y4K0 1/20 0.38
DPP4 P27487 3/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
CYP1A2 P05177 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
SCN4A P35499 2/20 0.34
AR P10275 3/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL8703025 1.00 TSHR (0.54) TSHRLOXL2DPP4MEN1MAPT
SCHEMBL1922926 0.82 TSHR (0.56) TSHRMEN1MAPTKMT2ANPSR1
SCHEMBL6351539 0.80 TSHR (0.54) TSHRMEN1MAPTKMT2ANPSR1
SCHEMBL6739582 0.80 TSHR (0.54) TSHRMEN1MAPTKMT2ANPSR1
SCHEMBL6740953 0.80 TSHR (0.54) TSHRMEN1MAPTKMT2ANPSR1
SCHEMBL394915 0.78 CYP1A2 (0.43) TSHRLOXL2DPP4TDP1CYP1A2
SCHEMBL29239979 0.78 PNMT (0.39) TSHRLOXL2DPP4MAPTCYP1A2
SCHEMBL28190550 0.78 CYP3A4 (0.44) TSHRLOXL2DPP4MEN1MAPT
SCHEMBL12490636 0.77 TSHR (0.50) TSHRMEN1MAPTKMT2ANPSR1
SCHEMBL28234295 0.77 TSHR (0.50) TSHRMEN1MAPTKMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036061-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2000-09-20 EP disclosed
WO-1999029664-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 1999-06-17 WO disclosed
US-5736568-A ANTIALLERGENS; IMMUNOMODULANTS KNOLL AKTIENGESELLSCHAFT (DE) 1998-04-07 US disclosed