SCHEMBL7359075

SCHEMBL7359075

CCOC(=O)[C@@H](Cc1ccc(-c2ccno2)cc1)NC

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2C19 P33261 1/20 0.42
EDNRB P24530 10/20 0.40
EDNRA P25101 10/20 0.40
KMT2A Q03164 3/20 0.40
ELANE P08246 1/20 0.39
CYP3A4 P08684 1/20 0.38
TP53 P04637 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359080 1.00 CYP2C9 (0.42) CYP2C9CYP1A2CYP2D6CYP19A1CYP2C19
SCHEMBL7229480 0.88 TACR1 (0.45) CYP2C9CYP1A2CYP2D6CYP19A1CYP2C19
SCHEMBL7437288 0.82 EDNRB (0.49) EDNRBEDNRATP53
SCHEMBL7361274 0.82 EDNRB (0.49) EDNRBEDNRATP53
SCHEMBL7365507 0.82 TPH1 (0.47) CYP2C9CYP1A2CYP2D6CYP19A1CYP2C19
SCHEMBL7360008 0.82 TPH1 (0.47) CYP2C9CYP1A2CYP2D6CYP19A1CYP2C19
SCHEMBL7445181 0.82 TPH1 (0.47) CYP2C9CYP1A2CYP2D6CYP19A1CYP2C19
SCHEMBL22240360 0.77 EPHX2 (0.52) CYP2C9CYP1A2CYP2C19KMT2AMEN1
SCHEMBL8246144 0.76 BACE1 (0.53) KMT2A
SCHEMBL973730 0.76 BACE1 (0.53) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997011960-A1 ANTAGONISTS OF ENDOTHELIN RECEPTORS JAPAT LTD. (CH) 1997-04-03 WO disclosed