SCHEMBL7361232

SCHEMBL7361232

N[C@H](CC1CCCCC1)C(O)C(=O)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 15/20 0.60
METAP1 P53582 7/20 0.57
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361364 0.86 METAP2 (0.60) METAP2METAP1
SCHEMBL14984996 0.85 METAP2 (0.47) METAP2METAP1MAPT
SCHEMBL7349858 0.85 METAP2 (0.68) METAP2METAP1
SCHEMBL7363265 0.84 METAP2 (0.57) METAP2METAP1
SCHEMBL25859126 0.83 METAP2 (0.45) METAP2METAP1MAPT
SCHEMBL12022078 0.83 METAP2 (0.45) METAP2METAP1MAPT
Hydrochloric Acid SCHEMBL7362363 0.83 METAP2 (0.56) METAP2METAP1
SCHEMBL19254379 0.82 METAP2 (0.44) METAP2METAP1MAPT
SCHEMBL7445063 0.81 METAP2 (0.78) METAP2METAP1
SCHEMBL7353275 0.81 METAP2 (0.60) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed