SCHEMBL7361595

SCHEMBL7361595

CCOC(=O)CC(O)Cc1cccc(C#N)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.48
CD274 Q9NZQ7 1/20 0.48
FFAR1 O14842 2/20 0.47
FOLH1 Q04609 1/20 0.45
CNR2 P34972 1/20 0.44
GLA P06280 1/20 0.43
NLRP3 Q96P20 1/20 0.42
DPP4 P27487 1/20 0.42
DPP7 Q9UHL4 1/20 0.42
MMP12 P39900 1/20 0.41
MMP13 P45452 1/20 0.41
PIN1 Q13526 1/20 0.41
MAOB P27338 1/20 0.41
POLB P06746 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
CYP1A2 P05177 1/20 0.40
GRM5 P41594 1/20 0.40
IDH1 O75874 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
FNTA P49354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23139004 0.83 FFAR1 (0.49) PDCD1CD274FFAR1FOLH1CNR2
SCHEMBL7360596 0.83 FFAR1 (0.49) PDCD1CD274FFAR1FOLH1CNR2
SCHEMBL7363960 0.82 PDCD1 (0.46) PDCD1CD274FFAR1FOLH1CNR2
SCHEMBL2673187 0.81 PDCD1 (0.49) PDCD1CD274FFAR1FOLH1CNR2
SCHEMBL30088453 0.81 PDCD1 (0.54) PDCD1CD274FFAR1CNR2GLA
SCHEMBL5725267 0.81 PDCD1 (0.54) PDCD1CD274FFAR1CNR2GLA
SCHEMBL7453413 0.80 FFAR1 (0.46) PDCD1CD274FFAR1FOLH1CNR2
SCHEMBL7360595 0.79 PDCD1 (0.50) PDCD1CD274FFAR1CNR2CYP1A2
SCHEMBL7403825 0.79 DPP7 (0.51) PDCD1CD274FFAR1FOLH1CNR2
SCHEMBL7404834 0.79 DPP7 (0.51) PDCD1CD274FFAR1FOLH1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed