SCHEMBL7360596

SCHEMBL7360596

CCOC(=O)C(O)Cc1cccc(C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.49
PDCD1 Q15116 1/20 0.48
CD274 Q9NZQ7 1/20 0.48
FOLH1 Q04609 1/20 0.48
GLA P06280 1/20 0.46
NLRP3 Q96P20 1/20 0.44
CNR2 P34972 1/20 0.44
MAOB P27338 1/20 0.43
POLB P06746 1/20 0.43
IDH1 O75874 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
CYP1A2 P05177 1/20 0.42
GRM5 P41594 1/20 0.42
MEP1A Q16819 1/20 0.42
MEP1B Q16820 1/20 0.42
FNTA P49354 1/20 0.42
FNTB P49356 1/20 0.42
SETD7 Q8WTS6 1/20 0.42
SCN8A Q9UQD0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23139004 1.00 FFAR1 (0.49) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL2673187 0.87 PDCD1 (0.49) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL19803700 0.87 NLRP3 (0.53) FFAR1FOLH1GLANLRP3MAOB
SCHEMBL7403825 0.85 DPP7 (0.51) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL7404834 0.85 DPP7 (0.51) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL7404836 0.85 DPP7 (0.51) FFAR1PDCD1CD274FOLH1GLA
Hydrochloric Acid SCHEMBL7403820 0.84 DPP7 (0.50) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL10707875 0.84 PDCD1 (0.46) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL7361595 0.83 PDCD1 (0.48) FFAR1PDCD1CD274FOLH1GLA
SCHEMBL20702757 0.81 FOLH1 (0.60) FFAR1FOLH1GLAMAOBFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111356680-B Selective inhibitors of NLRP3 inflammasome 诺瑟拉有限公司 2023-11-28 CN disclosed
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed