SCHEMBL7361718

SCHEMBL7361718

Cn1ccnc1C(O)C(N)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
MAPT P10636 1/20 0.51
CYP2D6 P10635 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.41
CSNK1E P49674 1/20 0.40
ADAM17 P78536 1/20 0.40
KMT2A Q03164 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.39
FGB P02675 1/20 0.39
ALOX15 P16050 1/20 0.39
TNNI3 P19429 1/20 0.39
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
BRCA1 P38398 1/20 0.39
TNNT2 P45379 1/20 0.39
CASP7 P55210 1/20 0.39
TNNC1 P63316 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15358494 0.83 KDM4E (0.61) KDM4EMAPTCYP2D6L3MBTL1KMT2A
SCHEMBL7318117 0.78 MAPT (0.41) MAPTCYP2D6KMT2ATDP1CYP1A2
SCHEMBL7361684 0.74 CSNK1E (0.40) CYP2D6CSNK1EALOX15MAPK1CASP1
SCHEMBL7393751 0.74 CSNK1E (0.42) CYP2D6CSNK1ETAAR1MAOASLC6A2
SCHEMBL11057220 0.72 KDM4E (0.48) KDM4EMAPTCYP2D6L3MBTL1KMT2A
SCHEMBL13919517 0.72 MAPT (0.65) KDM4EMAPTL3MBTL1KMT2AMEN1
SCHEMBL13257729 0.70
SCHEMBL950298 0.70 KDM4E (0.65) KDM4EMAPTCYP2D6L3MBTL1KMT2A
SCHEMBL30824582 0.70 KDM4E (0.65) KDM4EMAPTCYP2D6L3MBTL1KMT2A
SCHEMBL20569975 0.69 TDP1 (0.43) CYP2D6KMT2ATDP1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415981-A4 RETROVIRAL PROTEASE INHIBITORS 1991-10-09 EP disclosed
EP-0415981-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0342541-A2 Retroviral protease inhibitors ABBOTT LABORATORIES (US) 1989-11-23 EP disclosed
WO-1989010752-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed