SCHEMBL7361684

SCHEMBL7361684

Cn1nnnc1C(O)C(N)Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1E P49674 1/20 0.40
SLC6A2 P23975 5/20 0.39
SLC6A3 Q01959 4/20 0.39
SLC6A4 P31645 3/20 0.39
TAAR1 Q96RJ0 2/20 0.39
MAOA P21397 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CYP2A6 P11509 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
SLC15A1 P46059 1/20 0.38
EPHX1 P07099 1/20 0.37
CYP2D6 P10635 1/20 0.37
LAP3 P28838 3/20 0.36
ANPEP P15144 1/20 0.36
RNPEP Q9H4A4 1/20 0.36
DNPEP Q9ULA0 1/20 0.36
MAPK1 P28482 2/20 0.36
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361718 0.74 KDM4E (0.54) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL3700170 0.74 CNR2 (0.43) TAAR1CYP2D6ALDH1A1SMN1; SMN2
SCHEMBL7393751 0.74 CSNK1E (0.42) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL13919551 0.71 MAPT (0.53) MAOASIGMAR1LAP3SMN1; SMN2PKM
SCHEMBL27502071 0.69 EPHX1 (0.52) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL22885976 0.69 CYP1A2 (0.42) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL23752456 0.67 SLC6A2 (0.61) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL6193282 0.67 SLC6A2 (0.61) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL8091553 0.67 SLC6A2 (0.61) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1
SCHEMBL2232612 0.67 SLC6A2 (0.61) CSNK1ESLC6A2SLC6A3SLC6A4TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415981-A4 RETROVIRAL PROTEASE INHIBITORS 1991-10-09 EP disclosed
EP-0415981-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0342541-A2 Retroviral protease inhibitors ABBOTT LABORATORIES (US) 1989-11-23 EP disclosed
WO-1989010752-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed