SCHEMBL7361746

SCHEMBL7361746

COc1ccccc1NC(=O)C(O)[C@H](N)CC1CCCCC1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 11/20 0.64
METAP1 P53582 6/20 0.64
TDP1 Q9NUW8 3/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.54
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362176 0.90 METAP2 (0.58) METAP2METAP1TDP1L3MBTL1
Hydrochloric Acid SCHEMBL7360639 0.89 METAP2 (0.58) METAP2METAP1TDP1L3MBTL1
SCHEMBL7354412 0.89 METAP2 (0.61) METAP2METAP1TDP1L3MBTL1SMN1; SMN2
Hydrochloric Acid SCHEMBL7356761 0.88 METAP2 (0.60) METAP2METAP1TDP1L3MBTL1SMN1; SMN2
SCHEMBL7359630 0.87 METAP2 (0.71) METAP2METAP1L3MBTL1SMN1; SMN2
SCHEMBL7355975 0.87 METAP2 (0.61) METAP2METAP1TAS1R3TAS1R1
SCHEMBL7353356 0.87 METAP2 (0.56) METAP2METAP1TDP1L3MBTL1
Hydrochloric Acid SCHEMBL7359061 0.86 METAP2 (0.60) METAP2METAP1TSHRTAS1R3TAS1R1
SCHEMBL7359902 0.86 METAP2 (0.60) METAP2METAP1TDP1L3MBTL1
SCHEMBL7362128 0.86 METAP2 (0.56) METAP2METAP1L3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US claimed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP claimed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO claimed
US-6242494-B1 ANGIOGENESIS INHIBITORS, ANTITUMOR AGENTS, DIABETIC RETINOPATHY, AND ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES 2001-06-05 US disclosed
EP-1073633-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 2001-02-07 EP disclosed
WO-1999057098-A2 SUBSTITUTED BETA-AMINO ACID INHIBITORS OF METHIONINE AMINOPEPTIDASE-2 ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed