SCHEMBL7361905

SCHEMBL7361905

CC(C)(C)OC(=O)N[C@@H](CC(=O)NCCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.55
KLK7 P49862 2/20 0.55
CACNA1B Q00975 5/20 0.49
CTSS P25774 4/20 0.49
SYK P43405 1/20 0.49
PPARA Q07869 1/20 0.49
ACE P12821 1/20 0.48
CTSK P43235 4/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
MAPT P10636 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9223452 0.93 CTSS (0.53) KLK5KLK7CTSSSYKPPARA
SCHEMBL16574592 0.90 KLK5 (0.57) KLK5KLK7CACNA1BCTSSSYK
SCHEMBL23374042 0.87 KLK7 (0.49) KLK5KLK7CACNA1BCTSSSYK
SCHEMBL25715928 0.87 PPARA (0.56) KLK5KLK7CACNA1BCTSSSYK
SCHEMBL4370045 0.86 KLK5 (0.65) KLK5KLK7CACNA1BCTSSSYK
SCHEMBL7308756 0.86 MAPT (0.50) KLK5KLK7CTSSSYKPPARA
SCHEMBL9217565 0.86 MAPT (0.50) KLK5KLK7CTSSSYKPPARA
SCHEMBL3817109 0.84 PPARA (0.55) KLK5KLK7CACNA1BCTSSSYK
SCHEMBL1517760 0.84 PPARA (0.55) KLK5KLK7CACNA1BCTSSSYK
SCHEMBL16290229 0.84 PPARA (0.57) KLK5KLK7CTSSSYKPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed