SCHEMBL7361915

SCHEMBL7361915

COC(=O)C(Cc1cccc(C#N)c1)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.48
FOLH1 Q04609 1/20 0.46
GPR34 Q9UPC5 1/20 0.45
FFAR1 O14842 2/20 0.45
PIN1 Q13526 1/20 0.44
MAOB P27338 1/20 0.44
LMNA P02545 1/20 0.44
FFAR4 Q5NUL3 1/20 0.44
PPIA P62937 1/20 0.43
PSMB5 P28074 1/20 0.41
VNN1 O95497 1/20 0.41
GLA P06280 1/20 0.41
ADAMTS4 O75173 1/20 0.41
MMP13 P45452 1/20 0.41
MEP1A Q16819 1/20 0.41
MEP1B Q16820 1/20 0.41
ANPEP P15144 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361748 0.83 FFAR1 (0.46) NLRP3FOLH1GPR34FFAR1MAOB
SCHEMBL28851016 0.83 PSMB5 (0.54) PSMB5
SCHEMBL28851015 0.83 PSMB5 (0.54) PSMB5
SCHEMBL7527410 0.81 FFAR1 (0.48) NLRP3GPR34FFAR1MAOBLMNA
SCHEMBL5043134 0.79 NLRP3 (0.53) NLRP3FOLH1FFAR1PIN1MAOB
SCHEMBL19803700 0.79 NLRP3 (0.53) NLRP3FOLH1FFAR1PIN1MAOB
SCHEMBL2822759 0.78 DPP7 (0.52) NLRP3FOLH1PIN1MAOBLMNA
SCHEMBL8954810 0.78 DPP7 (0.52) NLRP3FOLH1PIN1MAOBLMNA
SCHEMBL6164203 0.78 DPP7 (0.52) NLRP3FOLH1PIN1MAOBLMNA
SCHEMBL21016636 0.78 NLRP3 (0.46) NLRP3FOLH1FFAR1PIN1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed