SCHEMBL7362380

SCHEMBL7362380

CC(C)(C)OC(=O)NC(Cc1ccccc1)C(C=CC(=O)O)O[Si](C)(C)C(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.47
CTSS P25774 4/20 0.47
CTSK P43235 3/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
ATM Q13315 1/20 0.46
ACE P12821 1/20 0.45
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
PKM P14618 2/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 1/20 0.43
ALOX15 P16050 1/20 0.43
XBP1 P17861 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9657327 1.00 KLK5 (0.47) KLK5CTSSCTSKCTSLCTSB
SCHEMBL9658726 0.88 KLK5 (0.49) KLK5CTSSCTSKCTSLCTSB
SCHEMBL9659473 0.88 ATM (0.51) KLK5CTSSCTSKCTSLCTSB
SCHEMBL3053578 0.84 ACE (0.43) KLK5CTSSCTSKCTSLCTSB
SCHEMBL3053580 0.84 ACE (0.43) KLK5CTSSCTSKCTSLCTSB
SCHEMBL3045572 0.83 KLK5 (0.42) KLK5CTSSCTSKCTSLCTSB
SCHEMBL3045577 0.83 KLK5 (0.42) KLK5CTSSCTSKCTSLCTSB
SCHEMBL9657554 0.82 KLK5 (0.48) KLK5CTSSCTSKCTSLCTSB
SCHEMBL9657551 0.82 KLK5 (0.48) KLK5CTSSCTSKCTSLCTSB
SCHEMBL9659720 0.81 KLK5 (0.55) KLK5CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130468-A Process for the preparation of a dipeptide isostere ABBOTT LABORATORIES (US) 1992-07-14 US disclosed
EP-0415981-A4 RETROVIRAL PROTEASE INHIBITORS 1991-10-09 EP disclosed
EP-0415981-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0342541-A2 Retroviral protease inhibitors ABBOTT LABORATORIES (US) 1989-11-23 EP disclosed
WO-1989010752-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed