SCHEMBL7362629

SCHEMBL7362629

COc1ccc(NC(=O)c2c[nH]c3c2C(=O)NCC3)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.43
RAB9A P51151 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
NPC1 O15118 3/20 0.43
GAA P10253 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
MAOB P27338 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
DHODH Q02127 4/20 0.41
JMJD7 P0C870 1/20 0.40
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
GPR35 Q9HC97 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7397673 0.89 POLB (0.40) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL7359461 0.84 DHODH (0.44) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL7400116 0.84 DHODH (0.47) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL6778783 0.82 ABCB1 (0.42) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL7395738 0.82 ROCK2 (0.47) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL6768007 0.80 ABCB1 (0.43) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL6768158 0.79 SMN1; SMN2 (0.45) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL7449564 0.78 TP53 (0.46) ABCB1RAB9ASMN1; SMN2NPC1GAA
SCHEMBL7358902 0.76 TP53 (0.40) ABCB1RAB9ASMN1; SMN2NPC1DHODH
SCHEMBL7398344 0.76 DHODH (0.40) ABCB1RAB9ASMN1; SMN2NPC1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750702-A Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands NEUROGEN CORPORATION (US) 1998-05-12 US claimed
WO-1998002420-A9 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS 1998-04-23 WO claimed
WO-1998002420-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO claimed
US-5925770-A GAMMA-AMINOBUTYRIC ACID DERIVATIVES FOR DIAGNOSIS OR TREATMENT OF ANXIETY, SLEEP DISORDERS, SEIZURES, OVERDOSES OF BENZODIAZEPINE TYPE DRUGS, COGNITION ACTIVATORS NEUROGEN CORPORATION (US) 1999-07-20 US disclosed
US-5750702-A Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands NEUROGEN CORPORATION (US) 1998-05-12 US disclosed
WO-1998002420-A9 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS 1998-04-23 WO disclosed
WO-1998002420-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO disclosed