SCHEMBL7363360

SCHEMBL7363360

COc1ccc(C(C)C(=O)N2CCCC2C(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.49
ACE P12821 7/20 0.49
REN P00797 3/20 0.49
KDM4E B2RXH2 1/20 0.49
F2 P00734 1/20 0.49
LMNA P02545 1/20 0.49
LTA4H P09960 1/20 0.49
MAPT P10636 1/20 0.49
PEPD P12955 1/20 0.49
ALOX15 P16050 1/20 0.49
PTGS1 P23219 1/20 0.49
HTR2A P28223 1/20 0.49
PTGS2 P35354 1/20 0.49
HRH1 P35367 1/20 0.49
THPO P40225 1/20 0.49
PMP22 Q01453 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ACE2 Q9BYF1 1/20 0.49
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6783107 0.91 ACE (0.57) ACERENKDM4EF2LMNA
SCHEMBL6783112 0.91 ACE (0.57) ACERENKDM4EF2LMNA
SCHEMBL10173234 0.85 ACE (0.55) ACERENKDM4EF2LMNA
SCHEMBL9362237 0.85 ACE (0.55) ACERENKDM4EF2LMNA
SCHEMBL10173273 0.85 ACE (0.55) ACERENKDM4EF2LMNA
SCHEMBL3470058 0.80 ACE (0.56) NPSR1ACEACE2ALDH1A1
SCHEMBL6437755 0.79 DPP4 (0.69) ACE
SCHEMBL6437757 0.79 DPP4 (0.69) ACE
SCHEMBL24668844 0.79 ACE (0.52) NPSR1ACERENKDM4EF2
SCHEMBL4001869 0.79 ALDH1A1 (0.74) NPSR1LMNAALDH1A1SMN1; SMN2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165508-A1 ANTICANCER CALCIUM CHANNEL BLOCKERS Gray, Lloyd S. (US) 2002-01-02 EP disclosed
WO-2000059882-A1 ANTICANCER CALCIUM CHANNEL BLOCKERS GRAY LLOYD S (US) 2000-10-12 WO disclosed