SCHEMBL7363635

SCHEMBL7363635

Cc1cc(SC2=C(O)CC(CCc3ccsc3)(C(C)C)OC2=O)c(C(C)(C)C)cc1NS(=O)(=O)c1ccc(C(F)(F)F)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLNR O43193 1/20 0.42
NR1I2 O75469 1/20 0.42
ABCB11 O95342 1/20 0.42
PGR P06401 1/20 0.42
CTSD P07339 1/20 0.42
CHRM2 P08172 1/20 0.42
ADRA2A P08913 1/20 0.42
PGA5 P0DJD9 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
CTSE P14091 1/20 0.42
GABRA1 P14867 1/20 0.42
ADRA2C P18825 1/20 0.42
DRD1 P21728 1/20 0.42
HTR2A P28223 1/20 0.42
AGTR1 P30556 1/20 0.42
CCKAR P32238 1/20 0.42
ADRA1A P35348 1/20 0.42
PTGS2 P35354 1/20 0.42
PPARG P37231 1/20 0.42
OPRD1 P41143 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364625 0.90 MLNR (0.43) MLNRNR1I2ABCB11PGRCTSD
SCHEMBL6296570 0.80 LDHA (0.35) LDHALDHB
SCHEMBL5880834 0.79 MLNR (0.36) MLNRNR1I2ABCB11PGRCTSD
SCHEMBL6296396 0.79 LDHA (0.33) LDHALDHB
SCHEMBL6303245 0.79 LDHA (0.33) LDHALDHB
SCHEMBL6296398 0.79 LDHA (0.33) LDHALDHB
SCHEMBL6296536 0.78 LDHA (0.33) LDHALDHB
SCHEMBL6298389 0.78 LDHA (0.33) LDHALDHB
SCHEMBL6302995 0.75 LDHA (0.34) LDHALDHB
SCHEMBL6296400 0.75 LDHA (0.32) LDHALDHB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112269-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-07-04 EP disclosed
WO-2000015634-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2000-03-23 WO disclosed