SCHEMBL7363734

SCHEMBL7363734

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cccc(C(=O)O)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.61
ADORA3 P0DMS8 1/20 0.61
CACNA1F O60840 4/20 0.56
CACNA1D Q01668 4/20 0.56
CACNA1S Q13698 4/20 0.56
CACNA1C Q13936 4/20 0.56
HIF1A Q16665 3/20 0.56
MEN1 O00255 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
KMT2A Q03164 2/20 0.56
MAPT P10636 2/20 0.56
TSHR P16473 2/20 0.56
LMNA P02545 1/20 0.56
POLB P06746 1/20 0.56
MAPK1 P28482 1/20 0.56
GPR55 Q9Y2T6 1/20 0.56
CYP2D6 P10635 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9150297 0.89 CACNA1B (0.71) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL28742846 0.87 CACNA1B (0.65) CACNA1B
SCHEMBL10659839 0.86 ADORA3 (0.55) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL27853207 0.85 TSHR (0.56) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7434340 0.84 ADORA3 (0.62) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL11783086 0.84 GAA (0.59) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL3905675 0.84 ADORA3 (0.83) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL11783074 0.83 GAA (0.64) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL10540800 0.83 ADORA3 (0.60) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7267420 0.83 CACNA1B (0.68) CACNA1BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378718-A Cardiovascular activity, hypotensive CEDONA PHARMACEUTICALS B.V. (NL) 1995-01-03 US disclosed
EP-0541634-A1 1,4-DIHYDROPYRIDINE DERIVATIVES CEDONA PHARMACEUTICALS B.V. (NL) 1993-05-19 EP disclosed
WO-1992002503-A1 NOVEL 1,4-DIHYDROPYRIDINE DERIVATIVES CEDONA PHARMACEUTICALS BV (NL) 1992-02-20 WO disclosed