SCHEMBL7364155

SCHEMBL7364155

Cc1cc(-c2cccc(C(F)(F)F)c2)n2ncc(C(=O)c3ccccc3)c2n1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.53
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
BRAF P15056 5/20 0.47
HSD17B10 Q99714 5/20 0.46
HPGD P15428 3/20 0.46
TSHR P16473 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
ALDH1A1 P00352 4/20 0.45
MAPK1 P28482 2/20 0.45
STAT1 P42224 1/20 0.45
CNR2 P34972 1/20 0.45
GLA P06280 1/20 0.44
LRRK2 Q5S007 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362761 0.87 MAPT (0.61) KDM4EMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL7360041 0.83 KDM4E (0.75) KDM4EBRAF
SCHEMBL7364602 0.82 MAPT (0.52) KDM4EMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL7364096 0.81 MAPT (0.53) KDM4EMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL7361109 0.76 KDM4E (0.74) KDM4EBRAF
SCHEMBL9468353 0.75 KDM4E (0.70) KDM4EMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL7362754 0.75 KDM4E (0.68) KDM4EBRAF
SCHEMBL10941469 0.75 MAPT (0.52) KDM4EMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL7369441 0.75 KDM4E (0.71) KDM4EBRAF
SCHEMBL7370603 0.75 KDM4E (0.67) KDM4EBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed