SCHEMBL7364258

SCHEMBL7364258

NC(=O)c1ccccc1-n1ccnc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.57
CYP3A4 P08684 7/20 0.52
CYP1A2 P05177 4/20 0.52
CYP2D6 P10635 4/20 0.52
CYP2C19 P33261 4/20 0.52
MAPK1 P28482 2/20 0.52
CYP2C9 P11712 3/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
MAPT P10636 1/20 0.49
PMP22 Q01453 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
TBXAS1 P24557 1/20 0.48
GAA P10253 2/20 0.46
NPC1 O15118 1/20 0.46
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
BAZ2B Q9UIF8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10438238 0.98 IDO1 (0.56) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL726313 0.85 IDO1 (0.59) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL5319528 0.84 IDO1 (0.47) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL13739921 0.84 CYP3A4 (0.48) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL7231541 0.83 IDO1 (0.57) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL6601781 0.83 IDO1 (0.57) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL1132341 0.83 IDO1 (0.57) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL15881145 0.82 SIRT3 (0.49) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL11802077 0.81 CYP19A1 (0.56) IDO1CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL1239412 0.81 IDO1 (0.54) IDO1CYP3A4CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249692-B 2-imidazole benzamide active compound for preventing and treating wheat take-all and wheat stem basal rot 河南农业大学 2024-01-30 CN claimed
WO-2014111871-A1 4,5-DIHYDROISOXAZOLE DERIVATIVES AS NAMPT INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2014-07-24 WO claimed
EP-2691375-A1 SUBSTITUTED BENZIMIDAZOLES Bayer Intellectual Property GmbH (DE) 2014-02-05 EP claimed
WO-2012130905-A1 SUBSTITUTED BENZIMIDAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-04 WO claimed
CN-114249692-B 2-imidazole benzamide active compound for preventing and treating wheat take-all and wheat stem basal rot 河南农业大学 2024-01-30 CN disclosed
CN-114249692-B 2-imidazole benzamide active compound for preventing and treating wheat take-all and wheat stem basal rot 河南农业大学 2024-01-30 CN disclosed
WO-2015055994-A1 CYCLOPENTYLBENZAMIDE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF PSYCHOTIC AND COGNITIVE DISORDERS TAKEDA CAMBRIDGE LIMITED (GB) 2015-04-23 WO disclosed
CN-1900080-A Inhibitors of cruzipain and other cysteine proteases AMURA THERAPEUTICS LTD (GB) 2007-01-24 CN disclosed
CN-1269822-C Inhibitors of kruenza protease and other cysteine proteases AMURA THERAPEUTICS LTD (GB) 2006-08-16 CN disclosed
WO-1996017630-A9 SUBSTITUTED BENZAMIDES AND RADIOLIGAND ANALOGS AND METHODS OF USE 1996-08-08 WO disclosed
WO-1996017630-A1 SUBSTITUTED BENZAMIDES AND RADIOLIGAND ANALOGS AND METHODS OF USE VANDERBILT UNIVERSITY (US) 1996-06-13 WO disclosed