SCHEMBL7364281

SCHEMBL7364281

CC(C)C[C@H](NCc1ccc(C(C)(C)C)cc1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.52
MME P08473 2/20 0.50
ACE P12821 2/20 0.50
CPA1 P15085 2/20 0.50
ACE2 Q9BYF1 2/20 0.50
IL1RN P18510 1/20 0.50
ERAP2 Q6P179 1/20 0.50
ERAP1 Q9NZ08 1/20 0.50
PSMB5 P28074 2/20 0.49
CACNA1B Q00975 2/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
KMT2A Q03164 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
PTPN1 P18031 1/20 0.47
CTSS P25774 3/20 0.46
CTSL P07711 1/20 0.46
CTSK P43235 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440191 0.90 KMT2A (0.52) MMEACECPA1ACE2MEN1
SCHEMBL7440200 0.90 KMT2A (0.52) MMEACECPA1ACE2MEN1
Hydrochloric Acid SCHEMBL7896063 0.89 KMT2A (0.51) MMEACECPA1ACE2MEN1
Hydrochloric Acid SCHEMBL7896068 0.89 KMT2A (0.51) MMEACECPA1ACE2MEN1
SCHEMBL7369252 0.89 REN (0.53) RENMMEACECPA1ACE2
SCHEMBL7405538 0.89 REN (0.53) RENMMEACECPA1ACE2
SCHEMBL8179352 0.88 MME (0.56) RENMMEACECPA1ACE2
SCHEMBL7408594 0.86 REN (0.56) RENMMEACECPA1ACE2
SCHEMBL7364989 0.86 MME (0.56) RENMMEACECPA1ACE2
SCHEMBL24206195 0.84 MME (0.48) RENMMEACECPA1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed