SCHEMBL7365754

SCHEMBL7365754

COc1ccc(CNC(=O)c2cc(C(F)(F)F)ccc2NC2CCC(OC(=O)c3ccccc3)CC2)cc1C#N

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 14/20 0.42
PPARG P37231 4/20 0.41
PPARD Q03181 5/20 0.40
PSEN1 P49768 3/20 0.40
PSEN2 P49810 3/20 0.40
APH1B Q8WW43 3/20 0.40
NCSTN Q92542 3/20 0.40
APH1A Q96BI3 3/20 0.40
PSENEN Q9NZ42 3/20 0.40
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
GPR6 P46095 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365758 1.00 PPARA (0.42) PPARAPPARGPPARDPSEN1PSEN2
SCHEMBL7370786 0.89 MRGPRX4 (0.44) PPARAPPARGPPARDPSEN1PSEN2
SCHEMBL7370784 0.89 MRGPRX4 (0.44) PPARAPPARGPPARDPSEN1PSEN2
SCHEMBL7365379 0.87 LMNA (0.41) PPARAPPARGPPARDKCNQ3KCNQ2
SCHEMBL7365381 0.87 LMNA (0.41) PPARAPPARGPPARDKCNQ3KCNQ2
SCHEMBL7367034 0.85 PPARA (0.44) PPARAPPARGPPARDPSEN1PSEN2
SCHEMBL7360754 0.77 PPARA (0.49) PPARAPPARGPPARDPSEN1PSEN2
SCHEMBL6940168 0.77 MAPT (0.46)
SCHEMBL6940165 0.77 MAPT (0.46)
SCHEMBL6940097 0.77 LMNA (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001030745-A1 ANTHRANILIC ACID DERIVATIVES AS INHIBITORS OF THE CGMP-PHOSPHODIESTERASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-03 WO disclosed