SCHEMBL7365839

SCHEMBL7365839

COc1ccc(C(=O)c2cnn3c(-c4cccnc4)ccnc23)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 1/20 0.50
PIM1 P11309 4/20 0.48
LIMK1 P53667 2/20 0.48
MAP2K1 Q02750 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
MAPK13 O15264 3/20 0.46
TLR8 Q9NR97 1/20 0.45
GSK3A P49840 3/20 0.44
AKT1 P31749 2/20 0.44
PIM3 Q86V86 2/20 0.44
DAPK3 O43293 1/20 0.44
MAPK9 P45984 1/20 0.44
NEK2 P51955 1/20 0.44
PLK3 Q9H4B4 1/20 0.44
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
EPHA2 P29317 1/20 0.41
MARK2 Q7KZI7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362153 0.88 KDM4E (0.64) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7360098 0.86 MAP2K1 (0.56) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7362717 0.84 TLR8 (0.55) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7366983 0.83 KDM4E (0.54) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7369092 0.83 KDM4E (0.65) KDM4EPIM1DYRK1BMAPK13TLR8
SCHEMBL7366580 0.82 MAP2K1 (0.55) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7361400 0.82 CLK4 (0.62) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7366385 0.81 MAP2K1 (0.49) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7369929 0.80 KDM4E (0.55) KDM4EALDH1A1PIM1LIMK1MAP2K1
SCHEMBL7363924 0.80 KDM4E (0.58) KDM4EALDH1A1PIM1LIMK1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed