SCHEMBL7366515

SCHEMBL7366515

COc1ccc(C(N)=O)c2[nH]cnc12

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.45
ABL1 P00519 1/20 0.42
RAD52 P43351 1/20 0.42
RIN1 Q13671 1/20 0.42
BRD4 O60885 4/20 0.41
NNMT P40261 2/20 0.40
BTK Q06187 2/20 0.39
AURKA O14965 1/20 0.39
RPS6KB1 P23443 1/20 0.39
QPCT Q16769 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
BRAF P15056 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20079235 0.85 ABL1 (0.42) ABL1RAD52RIN1BRD4QPCT
SCHEMBL18248868 0.82 GAA (0.47) PARP1ABL1RAD52RIN1BRD4
SCHEMBL14347857 0.80 PARP1 (0.49) PARP1NNMTBTKAURKA
SCHEMBL2272157 0.78 ABL1 (0.53) ABL1RAD52RIN1BRD4BRAF
SCHEMBL2273213 0.76 ABL1 (0.47) ABL1RAD52RIN1BRD4
SCHEMBL29579061 0.75 BRD4 (0.40) PARP1ABL1RAD52RIN1BRD4
SCHEMBL8575388 0.74 PTGS1 (0.44) ABL1RAD52RIN1BRD4QPCT
SCHEMBL13448012 0.73 ABL1 (0.49) ABL1RAD52RIN1BRD4BRAF
SCHEMBL14348180 0.73 PARP1 (0.53) PARP1NNMTRPS6KB1
SCHEMBL22533636 0.73 PARP1 (0.56) PARP1BRD4NNMTQPCTMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934307-A1 SUBSTITUTED AZABICYLIC COMPOUNDS AND THEIR USE AS INHIBITORS OF THE PRODUCTION OF TNF AND CYCLIC AMP PHOSPHODIESTERASE RHONE-POULENC RORER LIMITED (GB) 1999-08-11 EP claimed
WO-1997048697-A1 SUBSTITUTED AZABICYLIC COMPOUNDS AND THEIR USE AS INHIBITORS OF THE PRODUCTION OF TNF AND CYCLIC AMP PHOSPHODIESTERASE RHONE-POULENC RORER LIMITED (GB) 1997-12-24 WO claimed
EP-0934307-A1 SUBSTITUTED AZABICYLIC COMPOUNDS AND THEIR USE AS INHIBITORS OF THE PRODUCTION OF TNF AND CYCLIC AMP PHOSPHODIESTERASE RHONE-POULENC RORER LIMITED (GB) 1999-08-11 EP disclosed
WO-1997048697-A1 SUBSTITUTED AZABICYLIC COMPOUNDS AND THEIR USE AS INHIBITORS OF THE PRODUCTION OF TNF AND CYCLIC AMP PHOSPHODIESTERASE RHONE-POULENC RORER LIMITED (GB) 1997-12-24 WO disclosed