SCHEMBL7366871

SCHEMBL7366871

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCC(N(C)C)CC2)ccc1NC(=O)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.44
AVPR2 P30518 1/20 0.43
AVPR1A P37288 1/20 0.43
AVPR1B P47901 1/20 0.43
ADRA1D P25100 4/20 0.41
ADRA1A P35348 4/20 0.41
ADRA1B P35368 4/20 0.41
YAP1 P46937 2/20 0.39
PLK1 P53350 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TP53 P04637 1/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7342434 0.95 AVPR2 (0.42) CCR8AVPR2AVPR1AAVPR1BYAP1
SCHEMBL7370102 0.92 MEN1 (0.45) CCR8ADRA1DADRA1AADRA1BPLK1
SCHEMBL7339114 0.91 AVPR2 (0.42) AVPR2AVPR1AAVPR1BADRA1DADRA1A
SCHEMBL7339652 0.89 AVPR2 (0.42) CCR8AVPR2AVPR1AAVPR1BALDH1A1
SCHEMBL7781259 0.89 NPC1 (0.42) KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL7778279 0.87 AVPR2 (0.47) AVPR2AVPR1AAVPR1BMAPTMEN1
SCHEMBL7338105 0.86 AVPR2 (0.42) AVPR2AVPR1AAVPR1BADRA1DADRA1A
SCHEMBL7343158 0.86 AVPR2 (0.46) AVPR2AVPR1AAVPR1BMAPTTP53
SCHEMBL7336278 0.86 AVPR2 (0.48) AVPR2AVPR1AAVPR1BKDM4EMEN1
Hydrochloric Acid SCHEMBL7336979 0.85 AVPR2 (0.40) CCR8AVPR2AVPR1AAVPR1BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed