SCHEMBL7339114

SCHEMBL7339114

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCC(N(C)C)CC2)ccc1NC(=O)c1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.42
AVPR1A P37288 3/20 0.42
AVPR1B P47901 3/20 0.42
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
LMNA P02545 2/20 0.37
NPC1 O15118 1/20 0.37
AHR P35869 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 1/20 0.36
PLK1 P53350 2/20 0.36
POLB P06746 1/20 0.35
LRRK2 Q5S007 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339652 0.94 AVPR2 (0.42) AVPR2AVPR1AAVPR1BALDH1A1LMNA
SCHEMBL7339871 0.91 ALDH1A1 (0.39) AVPR2AVPR1AAVPR1BALDH1A1HPGD
SCHEMBL7366871 0.91 CCR8 (0.44) AVPR2AVPR1AAVPR1BALDH1A1SMN1; SMN2
SCHEMBL7778279 0.90 AVPR2 (0.47) AVPR2AVPR1AAVPR1BNPC1RAB9A
SCHEMBL7342434 0.88 AVPR2 (0.42) AVPR2AVPR1AAVPR1BALDH1A1HPGD
SCHEMBL7343093 0.88 POLB (0.39) AVPR2AVPR1AAVPR1BALDH1A1HPGD
SCHEMBL7343158 0.88 AVPR2 (0.46) AVPR2AVPR1AAVPR1BLMNASMN1; SMN2
Hydrochloric Acid SCHEMBL7336979 0.87 AVPR2 (0.40) AVPR2AVPR1AAVPR1BALDH1A1LMNA
Hydrochloric Acid SCHEMBL7780759 0.87 AVPR2 (0.46) AVPR2AVPR1AAVPR1BLMNASMN1; SMN2
SCHEMBL7345237 0.87 AVPR2 (0.46) AVPR2AVPR1AAVPR1BLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
US-6054457-A Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-25 US disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed