SCHEMBL7366872

SCHEMBL7366872

Cc1cc(C(=O)N2Cc3ccccc3Nc3ncccc32)c(C)cc1NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 10/20 0.56
AVPR1A P37288 4/20 0.56
OXTR P30559 1/20 0.56
AKT1 P31749 4/20 0.42
ALDH1A1 P00352 1/20 0.41
IDH1 O75874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7336470 0.93 AVPR2 (0.52) AVPR2AVPR1AOXTRAKT1
SCHEMBL7335141 0.89 AVPR2 (0.54) AVPR2AVPR1AOXTRAKT1
SCHEMBL7333134 0.84 AVPR2 (0.57) AVPR2AVPR1AOXTRAKT1
SCHEMBL7343088 0.82 AVPR2 (0.48) AVPR2AVPR1AOXTRALDH1A1
SCHEMBL7336360 0.82 AVPR2 (0.61) AVPR2AVPR1A
SCHEMBL7338077 0.80 AVPR2 (0.77) AVPR2AVPR1AOXTRALDH1A1
SCHEMBL7335578 0.77 AVPR2 (0.57) AVPR2AVPR1AOXTRAKT1IDH1
SCHEMBL7344791 0.77 AVPR2 (0.59) AVPR2AVPR1AOXTR
SCHEMBL7341289 0.76 AVPR2 (0.62) AVPR2AVPR1A
SCHEMBL7342975 0.76 AVPR2 (0.45) AVPR2AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed