SCHEMBL7367320

SCHEMBL7367320

COC(=O)CC1C(=O)N(C(C=O)OC(C)(C)C)CCN1C(=O)[C@H](CC(=O)OCc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 2/20 0.45
KLK7 P49862 1/20 0.45
CTSL P07711 1/20 0.41
CMA1 P23946 2/20 0.40
ACE P12821 1/20 0.40
CACNA1B Q00975 5/20 0.39
KMT2A Q03164 2/20 0.38
F2 P00734 1/20 0.37
PRSS1 P07477 1/20 0.37
CASP1 P29466 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367317 0.85 KLK7 (0.47) KLK5KLK7CTSLCMA1ACE
SCHEMBL7363006 0.85 KLK7 (0.47) KLK5KLK7CTSLCMA1ACE
SCHEMBL7363004 0.85 KLK7 (0.47) KLK5KLK7CTSLCMA1ACE
SCHEMBL7363000 0.85 KLK7 (0.47) KLK5KLK7CTSLCMA1ACE
SCHEMBL7367319 0.85 KLK7 (0.47) KLK5KLK7CTSLCMA1ACE
SCHEMBL29131321 0.75 ACE (0.65) KLK5KLK7CTSLCMA1ACE
SCHEMBL29131320 0.75 ACE (0.65) KLK5KLK7CTSLCMA1ACE
SCHEMBL7533944 0.75 ACE (0.65) KLK5KLK7CTSLCMA1ACE
SCHEMBL16510913 0.73 KLK7 (0.57) KLK5KLK7CTSLCACNA1BKMT2A
SCHEMBL3548960 0.73 PREP (0.67) KLK5KLK7CTSLCMA1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed