SCHEMBL7367568

SCHEMBL7367568

COc1ccc(C(=O)c2ccc(O)c(OC)c2)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 1/20 0.83
SLC22A8 Q8TCC7 1/20 0.83
ALDH1A1 P00352 1/20 0.75
GAA P10253 1/20 0.75
TUBB4A P04350 2/20 0.68
TUBB P07437 2/20 0.68
TUBA3C P0DPH7 2/20 0.68
TUBA1B P68363 2/20 0.68
TUBA4A P68366 2/20 0.68
TUBB4B P68371 2/20 0.68
TUBB3 Q13509 2/20 0.68
TUBB2A Q13885 2/20 0.68
TUBB8 Q3ZCM7 2/20 0.68
TUBA3E Q6PEY2 2/20 0.68
TUBA1A Q71U36 2/20 0.68
TUBA1C Q9BQE3 2/20 0.68
TUBB6 Q9BUF5 2/20 0.68
TUBB2B Q9BVA1 2/20 0.68
TUBB1 Q9H4B7 2/20 0.68
MEN1 O00255 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15814046 0.91 SLC22A6 (1.00) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL28149671 0.88 SLC22A6 (0.86) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL30355063 0.88 SLC22A6 (0.86) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL7373760 0.86 SLC22A6 (0.83) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL1545793 0.86 SLC22A6 (0.83) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL4818731 0.86 ALDH1A1 (1.00) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL7369813 0.86 SLC22A6 (0.89) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL10421110 0.85 SLC22A6 (0.80) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL7371991 0.85 SLC22A6 (0.80) SLC22A6SLC22A8ALDH1A1GAATUBB4A
SCHEMBL7374991 0.85 SLC22A6 (0.80) SLC22A6SLC22A8ALDH1A1GAATUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705703-A ENZYME INHIBITORS OF TRANSFERASES HOFFMANN-LA ROCHE INC. (US) 1998-01-06 US disclosed
US-5633371-A ENZYME INHIBITORS; TREATMENT OF DEPRESSION AND PARKINSON*S DISEASE HOFFMANN-LA ROCHE INC. (US) 1997-05-27 US disclosed
US-5476875-A Catechol derivatives HOFFMAN-LA ROCHE INC. (US) 1995-12-19 US disclosed
US-5389653-A Inhibitors of the enzyme catechol-O-methyltransferase; useful as co-medication in treatment of Parkinson's disease HOFFMAN-LA ROCHE INC. (US) 1995-02-14 US disclosed
EP-0442068-B1 Benzophenone derivatives and polymers containing phenolic hydroxyl groups BAYER AG (DE) 1994-06-08 EP disclosed
US-5236952-A Inhibit the enzyme catechol-O-methyltransferase; for treatment of Parkinson's disease administered with L-dopa HOFFMANN-LA ROCHE INC. (US) 1993-08-17 US disclosed
EP-0237929-B1 3,5-DISUBSTITUTED PYROCATECHOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-06-02 EP disclosed
EP-0442068-A2 Benzophenone derivatives and polymers containing phenolic hydroxyl groups BAYER AG (DE) 1991-08-21 EP disclosed
EP-0237929-A1 3,5-Disubstituted pyrocatechol derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-09-23 EP disclosed